CGP 52432

CAS No. 139667-74-6

CGP 52432 ( Cgp 52432; Cgp52432; Cgp52432 )

Catalog No. M17994 CAS No. 139667-74-6

CGP52432 is a very potent antagonist of GABAB receptors (IC50 = 85 nM).

Purity : 98%

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 43 In Stock
5MG 71 In Stock
10MG 129 In Stock
25MG 251 In Stock
50MG 437 In Stock
100MG 644 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    CGP 52432
  • Note
    Research use only, not for human use.
  • Brief Description
    CGP52432 is a very potent antagonist of GABAB receptors (IC50 = 85 nM).
  • Description
    Cgp 52432 is a GABA-A receptor antagonist
  • Synonyms
    Cgp 52432; Cgp52432; Cgp52432
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    GABAB
  • Research Area
    Neurological Disease
  • Indication
    ——

Chemical Information

  • CAS Number
    139667-74-6
  • Formula Weight
    384.23
  • Molecular Formula
    C15H24Cl2NO4P
  • Purity
    98%
  • Solubility
    DMSO : 5 mg/mL 13.01 mM;
  • SMILES
    CCOC(OCC)P(=O)(CCCNCC1=CC(=C(C=C1)Cl)Cl)O
  • Chemical Name
    Phosphinic acid, (3-(((3,4-dichlorophenyl)methyl)amino)propyl)(diethoxymethyl)-

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Bonanno G,etal.GABA(B) receptors as potential targets for drugs able to prevent excessive excitatory amino acid transmission in the spinal cord.Eur J Pharmacol. 1998 Dec 4;362(2-3):143-8.
molnova catalog
related products
  • LY392098

    LY392098 is a potentiator of AMPA receptor.

  • GDP366

    GDP366, induces cell growth inhibition, cellular senescence and mitotic catastrophe in human cancer cells. a dual inhibitor of survivin and Op18.

  • Citric acid monohydr...

    Citric Acid Monohydrate is a tricarboxylic acid found in citrus fruits. Citric acid is used as an excipient in pharmaceutical preparations due to its antioxidant properties. It maintains stability of active ingredients and is used as a preservative.