CGP 52432
CAS No. 139667-74-6
CGP 52432 ( Cgp 52432; Cgp52432; Cgp52432 )
Catalog No. M17994 CAS No. 139667-74-6
CGP52432 is a very potent antagonist of GABAB receptors (IC50 = 85 nM).
Purity : 98%
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
2MG | 43 | In Stock |
|
5MG | 71 | In Stock |
|
10MG | 129 | In Stock |
|
25MG | 251 | In Stock |
|
50MG | 437 | In Stock |
|
100MG | 644 | In Stock |
|
200MG | Get Quote | In Stock |
|
500MG | Get Quote | In Stock |
|
1G | Get Quote | In Stock |
|
Biological Information
-
Product NameCGP 52432
-
NoteResearch use only, not for human use.
-
Brief DescriptionCGP52432 is a very potent antagonist of GABAB receptors (IC50 = 85 nM).
-
DescriptionCgp 52432 is a GABA-A receptor antagonist
-
SynonymsCgp 52432; Cgp52432; Cgp52432
-
PathwayOthers
-
TargetOther Targets
-
RecptorGABAB
-
Research AreaNeurological Disease
-
Indication——
Chemical Information
-
CAS Number139667-74-6
-
Formula Weight384.23
-
Molecular FormulaC15H24Cl2NO4P
-
Purity98%
-
SolubilityDMSO : 5 mg/mL 13.01 mM;
-
SMILESCCOC(OCC)P(=O)(CCCNCC1=CC(=C(C=C1)Cl)Cl)O
-
Chemical NamePhosphinic acid, (3-(((3,4-dichlorophenyl)methyl)amino)propyl)(diethoxymethyl)-
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1.Bonanno G,etal.GABA(B) receptors as potential targets for drugs able to prevent excessive excitatory amino acid transmission in the spinal cord.Eur J Pharmacol. 1998 Dec 4;362(2-3):143-8.
molnova catalog
related products
-
NAV-2729
NAV-2729 inhibits six ArfGEFs (human ARNO, EFA6, BIG1, and BRAG2 and Legionella and Rickettsia RalF), the strongest effects being against BRAG2, Arf1 and Arf6.
-
Imipramine (hydrochl...
Imipramine (hydrochloride) is a first generation tricyclic antidepressant that acts primarily as an inhibitor of serotonin and norepinephrine transporters (Kds = 1.4 and 37 nM respectively).
-
2-Hydroxy atorvastat...
2-Hydroxy atorvastatin calcium salt is a hydroxy metabolite of Atorvastatin calcium salt which is a potent HMG-CoA reductase inhibitor (IC50 = 8 nM).